Study of the antitumour effects and the modulation of immune response by histamine in breast cancer

Abstract: Background: The aim of this work was to improve the knowledge of the role of histamine in breast cancer by assessing the therapeutic efficacy of histamine and histamine H4 receptor (H4R) ligands in a triple-negative breast cancer (TNBC) model developed in immunocompetent hosts. By using...

Descripción completa

Guardado en:
Detalles Bibliográficos
Autores principales: Nicoud, Melisa Beatriz, Sterle, Helena Andrea, Massari, Noelia A., Táquez Delgado, Mónica Alejandra, Formoso, Karina, Herrero Ducloux, María V., Martinel Lamas, Diego José, Cremaschi, Graciela A., Medina, Vanina Araceli
Formato: Artículo
Lenguaje:Inglés
Publicado: Nature 2022
Materias:
Acceso en línea:https://repositorio.uca.edu.ar/handle/123456789/14564
Aporte de:
id I33-R139-123456789-14564
record_format dspace
spelling I33-R139-123456789-145642023-11-23T17:03:42Z Study of the antitumour effects and the modulation of immune response by histamine in breast cancer Nicoud, Melisa Beatriz Sterle, Helena Andrea Massari, Noelia A. Táquez Delgado, Mónica Alejandra Formoso, Karina Herrero Ducloux, María V. Martinel Lamas, Diego José Cremaschi, Graciela A. Medina, Vanina Araceli CANCER DE MAMA TRIPLE NEGATIVO HISTAMINA RECEPTOR DE HISTAMINA H4 Abstract: Background: The aim of this work was to improve the knowledge of the role of histamine in breast cancer by assessing the therapeutic efficacy of histamine and histamine H4 receptor (H4R) ligands in a triple-negative breast cancer (TNBC) model developed in immunocompetent hosts. By using publicly available genomic data, we further investigated whether histidine decarboxylase (HDC) could be a potential biomarker. Methods: Tumours of 4T1 TNBC cells were orthotopically established in BALB/c mice. Treatments employed (mg kg−1): histamine (1 and 5), JNJ28610244 (H4R agonist, 1 and 5) and JNJ7777120 (H4R antagonist, 10). Results: Increased HDC gene expression is associated with better relapse-free and overall survival in breast cancer patients. Histamine treatment (5 mg kg−1) of 4T1 tumour-bearing mice reduced tumour growth and increased apoptosis. Although no immunomodulatory effects were observed in wild-type mice, significant correlations between tumour weight and cytotoxic lymphocyte infiltration were detected in H4R knockout mice. H4R agonist or antagonist differentially modulated tumour growth and immunity in 4T1 tumour-bearing mice. Conclusions: Histamine plays a complex role and stands out as a promising drug for TNBC treatment, which deserves to be tested in clinical settings. HDC expression level is associated with clinicopathological characteristics, suggesting a prognostic value in breast cancer. 2022-07-26T14:39:21Z 2022-07-26T14:39:21Z 2020 Artículo Nicoud, M. B. Study of the antitumour effects and the modulation of immune response by histamine in breast cancer [en línea]. British Journal of Cancer . 2020 (122). doi: https://doi.org/10.1038/s41416-019-0636-x. Disponible en: https://repositorio.uca.edu.ar/handle/123456789/14564 1532-1827 (online) 0007-0920 (impreso) https://repositorio.uca.edu.ar/handle/123456789/14564 10.1038/s41416-019-0636-x 31748740 eng Acceso abierto http://creativecommons.org/licenses/by-nc-sa/4.0/ application/pdf Nature British Journal of Cancer No.122., 2020
institution Universidad Católica Argentina
institution_str I-33
repository_str R-139
collection Repositorio Institucional de la Universidad Católica Argentina (UCA)
language Inglés
topic CANCER DE MAMA TRIPLE NEGATIVO
HISTAMINA
RECEPTOR DE HISTAMINA H4
spellingShingle CANCER DE MAMA TRIPLE NEGATIVO
HISTAMINA
RECEPTOR DE HISTAMINA H4
Nicoud, Melisa Beatriz
Sterle, Helena Andrea
Massari, Noelia A.
Táquez Delgado, Mónica Alejandra
Formoso, Karina
Herrero Ducloux, María V.
Martinel Lamas, Diego José
Cremaschi, Graciela A.
Medina, Vanina Araceli
Study of the antitumour effects and the modulation of immune response by histamine in breast cancer
topic_facet CANCER DE MAMA TRIPLE NEGATIVO
HISTAMINA
RECEPTOR DE HISTAMINA H4
description Abstract: Background: The aim of this work was to improve the knowledge of the role of histamine in breast cancer by assessing the therapeutic efficacy of histamine and histamine H4 receptor (H4R) ligands in a triple-negative breast cancer (TNBC) model developed in immunocompetent hosts. By using publicly available genomic data, we further investigated whether histidine decarboxylase (HDC) could be a potential biomarker. Methods: Tumours of 4T1 TNBC cells were orthotopically established in BALB/c mice. Treatments employed (mg kg−1): histamine (1 and 5), JNJ28610244 (H4R agonist, 1 and 5) and JNJ7777120 (H4R antagonist, 10). Results: Increased HDC gene expression is associated with better relapse-free and overall survival in breast cancer patients. Histamine treatment (5 mg kg−1) of 4T1 tumour-bearing mice reduced tumour growth and increased apoptosis. Although no immunomodulatory effects were observed in wild-type mice, significant correlations between tumour weight and cytotoxic lymphocyte infiltration were detected in H4R knockout mice. H4R agonist or antagonist differentially modulated tumour growth and immunity in 4T1 tumour-bearing mice. Conclusions: Histamine plays a complex role and stands out as a promising drug for TNBC treatment, which deserves to be tested in clinical settings. HDC expression level is associated with clinicopathological characteristics, suggesting a prognostic value in breast cancer.
format Artículo
author Nicoud, Melisa Beatriz
Sterle, Helena Andrea
Massari, Noelia A.
Táquez Delgado, Mónica Alejandra
Formoso, Karina
Herrero Ducloux, María V.
Martinel Lamas, Diego José
Cremaschi, Graciela A.
Medina, Vanina Araceli
author_facet Nicoud, Melisa Beatriz
Sterle, Helena Andrea
Massari, Noelia A.
Táquez Delgado, Mónica Alejandra
Formoso, Karina
Herrero Ducloux, María V.
Martinel Lamas, Diego José
Cremaschi, Graciela A.
Medina, Vanina Araceli
author_sort Nicoud, Melisa Beatriz
title Study of the antitumour effects and the modulation of immune response by histamine in breast cancer
title_short Study of the antitumour effects and the modulation of immune response by histamine in breast cancer
title_full Study of the antitumour effects and the modulation of immune response by histamine in breast cancer
title_fullStr Study of the antitumour effects and the modulation of immune response by histamine in breast cancer
title_full_unstemmed Study of the antitumour effects and the modulation of immune response by histamine in breast cancer
title_sort study of the antitumour effects and the modulation of immune response by histamine in breast cancer
publisher Nature
publishDate 2022
url https://repositorio.uca.edu.ar/handle/123456789/14564
work_keys_str_mv AT nicoudmelisabeatriz studyoftheantitumoureffectsandthemodulationofimmuneresponsebyhistamineinbreastcancer
AT sterlehelenaandrea studyoftheantitumoureffectsandthemodulationofimmuneresponsebyhistamineinbreastcancer
AT massarinoeliaa studyoftheantitumoureffectsandthemodulationofimmuneresponsebyhistamineinbreastcancer
AT taquezdelgadomonicaalejandra studyoftheantitumoureffectsandthemodulationofimmuneresponsebyhistamineinbreastcancer
AT formosokarina studyoftheantitumoureffectsandthemodulationofimmuneresponsebyhistamineinbreastcancer
AT herreroduclouxmariav studyoftheantitumoureffectsandthemodulationofimmuneresponsebyhistamineinbreastcancer
AT martinellamasdiegojose studyoftheantitumoureffectsandthemodulationofimmuneresponsebyhistamineinbreastcancer
AT cremaschigracielaa studyoftheantitumoureffectsandthemodulationofimmuneresponsebyhistamineinbreastcancer
AT medinavaninaaraceli studyoftheantitumoureffectsandthemodulationofimmuneresponsebyhistamineinbreastcancer
_version_ 1807949132658114560