Synthesis of 3β-hydroxy-5-cholenic acid from 3β-hydroxy-5-pregnen-20-one aimed at the preparation of labelled steroid compounds

3β-Hydroxy-5-cholenic acid was synthesized from 3β-hydroxy-5-pregnen-20-one in nine steps. The procedure would permit the labelling of C-22, C-23, and/or C-24 of the bile-acid side chain by choice of the appropriate labelled reagent. © 1977.

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Autor principal: Burton, G.
Otros Autores: Gros, E.G
Formato: Capítulo de libro
Lenguaje:Inglés
Publicado: 1977
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024 7 |2 cas  |a carbon, 7440-44-0; pregnenolone, 145-13-1; Carbon Radioisotopes; Cholenes; Pregnenolone, 145-13-1; Sterols 
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100 1 |a Burton, G. 
245 1 0 |a Synthesis of 3β-hydroxy-5-cholenic acid from 3β-hydroxy-5-pregnen-20-one aimed at the preparation of labelled steroid compounds 
260 |c 1977 
270 1 0 |m Gros, E.G.; Departamento de Quimica Orgánica, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires, Ciudad Universitaria, 1428 Buenos Aires, Argentina 
506 |2 openaire  |e Política editorial 
504 |a Ruzicka, Wettstein, Sexualhormone V. K�nstliche Herstellung des m�nnlichen Sexualhormons trans-Dehydro-androsteron und des Androsten-3,17-dions (1935) Helvetica Chimica Acta, 18, pp. 986-994 
504 |a Kučera, Šorm, Über steroide XXIX. Die isolierung von 3β-hydroxy-Δ5-nor-cholensäure und 3β-hydroxy-Δ5-cholestensäure-(26) aus den oxydationsprodukten des 3β-acetoxy-5α,6β-dibromcholestans mit chromtrioxyd (1958) Collection of Czechoslovak Chemical Communications, 23, pp. 116-124 
504 |a Riegel, Kaye, (1944) J. Am. chem. Soc., 66, pp. 723-724 
504 |a Meystre, Frey, Neher, Wettstein, Miescher, �ber Steroide. 48. Mitteilung. Ein einfacher Abbau der Gallens�uren-Seitenkette V. Die �berf�hrung von ?5-3 ?-Oxy-cholens�ure in Pregnenolon und Progesteron (1946) Helvetica Chimica Acta, 29, pp. 627-634 
504 |a Meystre, Wettstein, Miescher, �ber Steroide. (64. Mitteilung). Ein einfacher Abbau der Gallens�uren-Seitenkette VII. Weitere Wege zur Herstellung von Progesteron (1947) Helvetica Chimica Acta, 30, pp. 1022-1027 
504 |a Levin, Mclntosh, Jr., Spero, Rayman, Meinzer, (1948) J. Am. chem. Soc., 70, pp. 511-514 
504 |a Joly, Sauer, Bonner, Preparation of cholesterol-25-3H (1969) Journal of Labelled Compounds, 5, pp. 80-85 
504 |a Fieser, Fieser, (1959) Steroids, p. 509. , Reinhold, New York 
504 |a Bergstrom, Pääbo, Preparation of 3beta-Hydroxychol-5-enic Acid from Hyodesoxycholic Acid and Corresponding 24-14C-Labelled Acids. Bile Acids and Steroids 24. (1955) Acta Chemica Scandinavica, 9, pp. 699-701 
504 |a Porto, Baralle, Gros, (1972) J. steroid Biochem., 3, pp. 11-17 
504 |a Colonna, Gros, (1973) J. steroid Biochem., 4, pp. 171-179 
504 |a Chaudhuri, Williams, Nickolson, Gut, (1969) J. org. Chem., 34, pp. 3759-3766 
504 |a Scheineider, (1972) Tetrahedron, 28, pp. 2717-2726 
504 |a Narwid, Cooney, Uskokovic, (1974) Helv. chim. Acta, 57, pp. 771-781 
504 |a Faulkner, Stereoselective Synthesis of Trisubstituted Olefins (1971) Synthesis, pp. 175-189 
504 |a Letourneux, Lo, Chaudhuri, Gut, Acid-catalyzed rearrangement of 20-vinylpregn-5-ene-3.beta.,20-diol 3-acetate (1975) The Journal of Organic Chemistry, 40, pp. 516-518 
504 |a Sucrow, Inhaltsstoffe vonMomordica charantia L., I. Δ5.25-Stigmastadienol-(3β) und sein β-D-Glucosid (1966) Chemische Berichte, 99, pp. 2765-2777 
504 |a Dasgupta, Crump, Gut, (1974) J. org. Chem., 39, pp. 1658-1662 
504 |a Wicha, Bal, Synthesis of 25-hydroxycholesterol from 3?-hydroxyandrost-5-en-17-one. A method for stereospecific construction of a sterol side-chain (1975) Journal of the Chemical Society, Chemical Communications, pp. 968-969 
504 |a Monson, (1972) Advanced Organic Synthesis, p. 45. , Academic Press, New York 
504 |a Monson, (1972) Advanced Organic Synthesis, p. 140. , Academic Press, New York 
504 |a Hachey, Szczepanik, Berngruber, Klein, (1973) J. Label Compds., 9, pp. 703-719 
504 |a Porto, Gros, Synthesis of PREGN-5-en-3β-o1-20-one-20-14C (1968) Journal of Labelled Compounds, 4, pp. 276-278 
520 3 |a 3β-Hydroxy-5-cholenic acid was synthesized from 3β-hydroxy-5-pregnen-20-one in nine steps. The procedure would permit the labelling of C-22, C-23, and/or C-24 of the bile-acid side chain by choice of the appropriate labelled reagent. © 1977.  |l eng 
593 |a Departamento de Quimica Orgánica, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires, Ciudad Universitaria, 1428 Buenos Aires, Argentina 
650 1 7 |2 spines  |a CARBON 
690 1 0 |a CHOLANE DERIVATIVE 
690 1 0 |a PREGNENOLONE 
690 1 0 |a STEROL 
690 1 0 |a RADIOISOTOPE 
690 1 0 |a ARTICLE 
690 1 0 |a INFRARED SPECTROPHOTOMETRY 
690 1 0 |a ISOTOPE LABELING 
690 1 0 |a METHODOLOGY 
690 1 0 |a NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY 
690 1 0 |a OPTICAL ROTATION 
690 1 0 |a SYNTHESIS 
690 1 0 |a 3BETA HYDROXYCHOLENIC ACID 
690 1 0 |a IN VITRO STUDY 
690 1 0 |a STEROIDOGENESIS 
690 1 0 |a THEORETICAL STUDY 
690 1 0 |a CARBON RADIOISOTOPES 
690 1 0 |a CHOLENES 
690 1 0 |a ISOTOPE LABELING 
690 1 0 |a MAGNETIC RESONANCE SPECTROSCOPY 
690 1 0 |a OPTICAL ROTATION 
690 1 0 |a PREGNENOLONE 
690 1 0 |a SPECTROPHOTOMETRY, INFRARED 
690 1 0 |a STEROLS 
700 1 |a Gros, E.G. 
773 0 |d 1977  |g v. 8  |h pp. 69-72  |k n. 1  |p J. Steroid Biochem.  |x 00224731  |t Journal of Steroid Biochemistry 
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